PhI(OAc)2-mediated oxidative rearrangement of allylic amides: efficient synthesis of oxazoles and β-keto amides
文献信息
发布日期
2019-11-15
DOI
10.1039/C9QO01298B
影响因子
5.281
作者
Kang Xu, Shuang Yang, Zhenhua Ding
查看原文
摘要
A series of 2,5-disubstituted oxazoles and β-keto amides were synthesized from allylic amides via PhI(OAc)2-mediated intramolecular cyclization and oxidation with the migration of an aryl group. These reactions were performed under mild conditions with good functional group tolerance and gave the corresponding products in good to excellent yields.
期刊推荐
Physical Chemistry Chemical Physics
Environmental Toxicology and Pharmacology
Angewandte Chemie International Edition
Journal of Enzyme inhibition and Medicinal Chemistry
Journal of Medical Biochemistry
Advanced Engineering Materials
Current Pharmaceutical Biotechnology
Coloration Technology
Molecular Diversity
Molecules
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来源期刊
Organic Chemistry Frontiers
CiteScore:
7.8
自引率:
8.7%
年发文量:
724
Organic Chemistry Frontiers publishes high-quality research from across organic chemistry. Emphases are placed on studies that make significant contributions to the field of organic chemistry by reporting either new or significantly improved protocols or methodologies. Topics include, but are not limited to the following: Organic synthesis Development of synthetic methodologies Catalysis Natural products Functional organic materials Supramolecular and macromolecular chemistry Physical and computational organic chemistry
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